January 31, 2009
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We are grateful to OAKWOOD CHEMICAL for their generous support of Arkivoc and the FloHet Conferences - The Arkivoc Team
Recent Arkivoc Publications
Arkivoc 2008 Part (i): Special Issue 'Reviews and Accounts'
Syntheses of small cluster oligosaccharide mimetics (08-3623LU) [pp. 271-308]
Andreas H. Franz, Paul H. Gross and Vyacheslav V. Samoshin
Full Text: PDF (396K)
Arkivoc 2008 Part (xvii): General Papers
Synthesis, dynamic 1H NMR and theoretical study of aryl-nitrogen single bond rotational energy barriers in highly functionalized 4H-chromenes (08-3355CP) [pp. 12-19]
Roya Kabiri, Nourallah Hazeri, Sayyed Mostafa Habibi Khorassani, Malek Taher Maghsoodlou, Ali Ebrahimi, Lotfali Saghatforoush, Ghasem Marandi and Zahra Razmjoo
Full Text: PDF (369K)
Synthesis of DEFG ring system of cneorins (08-3570BP) [pp. 20-35]
Ari M. P. Koskinen and Ainoliisa J. Pihko
Full Text: PDF (354K)
Studies with 2-arylhydrazono-3-oxopropanals: Routes for the synthesis of pyridazine-3,4-dicarboxylate and 3,5-diaroyl pyrazoles (08-3518LP) [pp. 36-47]
Mariam A. Al-Shiekh, Hanady Y. Medrassi, Mohamed H. Elnagdi and Ebtisam A. Hafez
Full Text: PDF (2,809K)
Synthesis of symmetrical and unsymmetrical 1,3,4-oxadiazoles and their interconversion to 1,3,4-thiadiazoles and 1,2,4-triazoles (08-3538BP) [pp. 48-60]
Venkatapuram Padmavathi, Gali Sudhakar Reddy, Annaji Venkata Nagendra Mohan and Konda Mahesh
Full Text: PDF (245K)
Palladate salts from ionic liquids as catalysts in the Heck reaction (08-3535OP) [pp. 61-76]
Florence Gayet, Jean-Daniel Marty and Nancy Lauth-de Viguerie
Full Text: PDF (1,321K)
Convenient syntheses of new quinoline nucleosides bearing amino acid esters (08-3668LP) [pp. 77-89]
Ibrahim A. I. Ali
Full Text: PDF (257K)
Delocalized cationic azo dyes derived from 2-aminoselenazole-5-carbaldehyde (08-3408FP) [pp. 90-95]
Maria A. Salvador, Paulo Almeida, Lucinda V. Reis and Paulo F. Santos
Full Text: PDF (226K)
A study of conformational behaviour in some hexahydro-2H-isoxazolo[2,3-a]pyridines (08-3613LP) [pp. 96-106]
Shaikh A. Ali, Alaaeddin AlSbaiee and Mohamed I. M. Wazeer
Full Text: PDF (269K)
A convenient access to new pyrido[4,3-d]pyrimidine, thiazolo[3,4-c]pyrimidine and pyrimido[4,5-d]pyridazine derivatives (08-3561JP) [pp. 107-116]
Nabila A. Kheder, Yahia N. Mabkhot and Ahmad M. Farag
Full Text: PDF (236K)
Arylhydrazonals as aldehyde components in Baylis-Hillman reaction: synthesis of 5-hydroxy-2,3,4,5-tetrahydropyridazine-4-carbonitrile and 6,7,8,8a-tetrahydrocinnolin-5(1H)-one (08-3480AP) [pp. 117-121]
Ismail Abdelshafy Abdelhamid, Elham Sayed Darwish, Miead Adel Nasra, Fathy Mohamed Abdel-Gallil and Daisy Hanna Fleita
Full Text: PDF (260K)
New synthesis routes, characterization, electrochemical and spectral properties of p-substituted N-phenylpyrroles. Substituent effects (08-3340UP) [pp. 122-144]
A. K. D. Diaw, A. Yassar, D. Gningue-Sall and J.-J. Aaron
Full Text: PDF (555K)
Improving enantioselectivity via rationally tuning electronic effect of catalysts in the organocatalytic asymmetric aldol reaction (08-3567UP) [pp. 145-156]
Juanjuan Du, Zhiyi Li, Da-Ming Du and Jiaxi Xu
Full Text: PDF (304K)
Synthesis of liquid crystals derived from oxadiazole, isoxazole and tetrazole heterocycles (08-3409HP) [pp. 157-166]
Daniela Rubia dos Santos, Ana Gabriela Silva de Oliveira, Rafael Levi Coelho, Iêda Maria Begnini, Rachel Faverzani Magnago and Luciano da Silva
Full Text: PDF (185K)
One-pot synthesis of m-terphenyl-2'-carbaldehydes (08-3290MP) [pp. 167-172]
Bahaaldin Rashidzadeh, Farnaz Jafarpour and Akbar Saednya
Full Text: PDF (223K)
A facile synthesis, dynamic 1H NMR and theoretical study the novel stable heterocyclic phosphorus ylides containing tetrazole (08-3359HP) [pp. 173-183]
M. Amin Kazemian, Mahmoud Nassiri, Ali Ebrahimi, M. Taher Maghsoodlou, S. Mostafa Habibi-Khorassani and Fatemeh Vasheghani-Farahani
Full Text: PDF (377K)
Unexpected one-flask synthesis of 2,4-dialkylthiopentanedials via the reaction of alkylthioacetic aldehydes with dihalomethane and diethylamine (08-3641DP) [pp. 184-191]
Natalia A. Keiko, Ludmila G. Stepanova, Ekaterina A. Verochkina, Ludmila I. Larina and Yurii A. Chuvashev
Full Text: PDF (187K)
Ring transformation of chromone-3-carboxylic acid under nucleophilic conditions (08-3350MP) [pp. 192-204]
Magdy A. Ibrahim
Full Text: PDF (244K)
Synthesis of the first mixed-donor spiro-linked macrocyclic tetralactams (08-3609GP) [pp. 205-211]
Ahmed H. M. Elwahy, Hussni A. Muathen and Nour A. M. Aloweiny
Full Text: PDF (149K)
Efficient Niementowski synthesis of novel derivatives of 1,2,9,11-tetrasubstituted-7H-thieno[2',3':4,5]pyrimido[6,1-b]-quinazolin-7-one (08-3459MP) [pp. 212-220]
Sachin S. Laddha and Satayendra P. Bhatnagar
Full Text: PDF (219K)
Synthesis and antimicrobial activity of new Schiff bases containing coumarin moiety and their spectral characterization (08-3265MP) [pp. 221-233]
V. S. V. Satyanarayana, P. Sreevani, Amaravadi Sivakumar and V. Vijayakumar
Full Text: PDF (355K)
Oxazepines and thiazepines 46. Synthesis of tetracyclic 1,5-benzothiazepines by the reaction of α,β,γ,δ-unsaturated ketones with 2-aminothiophenol (08-3436NP) [pp. 234-240]
Albert Lévai and József Jekő
Full Text: PDF (193K)
Anhydrous zinc chloride: an efficient catalyst for one pot synthesis of 2,3,4,12-tetrahydrobenzothiazolo[2,3b]quinazolin-1-ones (08-3352AP) [pp. 241-247]
Satish A. Dake, Sunil U. Tekale, Swapnil R. Sarda, Wamanrao N. Jadhav, Sudhakar R. Bhusare and Rajendra P. Pawar
Full Text: PDF (155K)
Designer ligands. Part 14. Novel Mn(lI), Ni(II) and Zn(II) complexes of benzamide- and biphenyl-derived ligands (08-3568DP) [pp. 248-264]
Kevin W. Wellington, Perry T. Kaye and Gareth M. Watkins
Full Text: PDF (304K)
An efficient one-pot synthesis of dialkyl 8a-acetylamino-8-oxo-8,8a-dihydro-2H-1-oxacyclopenta[α]indene-2,3-dicarboxylate derivatives (08-3222MP) [pp. 265-272]
Mohammad Anary-Abbasinejad, Manouchehr Mazraeh-Seffid, Ehsanorreza Poorhassan, Alireza Hassanabadi and Forough Rastegari
Full Text: PDF (258K)
A practical synthesis and the pharmacological potency of gem-diphosphono substituted pyrimidines for treatment of bone resorption (08-3594HP) [pp. 273-286]
Azza A. Kamel and Maha D. Khidre
Full Text: PDF (302K)
Improved synthesis of the PAR-1 thrombine receptor antagonist RWJ-58259 (08-3630JP) [pp. 287-294]
Ángel M. Valdivielso, M. Teresa García-López and Rosario Herranz
Full Text: PDF (237K)
Supplementary Material: PDF (261K)
Arkivoc 2009 Part (ii): General Papers
A terminally modified pseudopeptide (Gly-m-aminobenzoic acid) produces supramolecular helix, staircase and water-mediated β-sheet through self-assembly (09-3501BP) [pp. 31-43]
Arpita Dutta, Sudeshna Kar, Roland Fröhlich, Pradyot Koley and Animesh Pramanik
Full Text: PDF (395K)
Solid state oxidative deprotection of 1,3-dithianes and 1,3-dithiolanes using poly(N,N'-dibromo-N-ethyl-benzene-1,3-disulfonamide) and N,N,N',N'-tetrabromobenzene-1,3-disulfonamide (09-3563LP) [pp. 44-51]
Ramin Ghorbani-Vaghei and Hojat Veisi
Full Text: PDF (278K)
Reusable silica supported poly phosphoric acid catalyzed three-component synthesis of 2H-indazolo[2,1-b]phthalazine-trione derivatives (09-3372NP) [pp. 59-67]
Hamid Reza Shaterian, Asghar Hosseinian and Majid Ghashang
Full Text: PDF (167K)
Arkivoc 2009 Part (vi): A Commemorative Issue in Honor of Prof. Henk C. van der Plas
Ring opening and ring expansion of 8-cyano-tetrazolo[1,5-a]pyridine with secondary amines. Reactions of azides, tetrazoles and nitrenes with nucleophiles, Part 2 (HP-3437MP) [pp. 30-37]
Chris Addicott, Paul V. Bernhardt and Curt Wentrup
Full Text: PDF (300K)
Synthesis of tetra- and pentacyclic carbazole-fused imides as potential antitumor agents (HP-3442MP) [pp. 38-47]
Norbert Haider, Rami Jbara, Johann Käferböck and Ursula Traar
Full Text: PDF (267K)
Synthesis and reactions of 1-amino-1,5,6,10b-tetrahydroimidazo[2,1-a]isoquinolin-2(3H)-ones (HP-3499MP) [pp. 48-62]
Joana Solovjova, Vytas Martynaitis, Wolfgang Holzer, Sven Mangelinckx, Norbert De Kimpe and Algirdas Šačkus
Full Text: PDF (323K)
Synthesis of 5-aryl-1-carboxyphenyl-3-(3-coumarinyl)-2-pyrazolines (HP-3695HP) [pp. 63-70]
Albert Lévai and József Jekő
Full Text: PDF (230K)
A first approach to 2,2’-bipyridine thiacrown ethers containing bisamide groups (HP-3465HP) [pp. 71-77]
Danuta Branowska, Justyna Ławecka, Waldemar Wysocki and Andrzej Rykowski
Full Text: PDF (657K)
Arkivoc 2009 Part (viii): A Commemorative Issue in Honor of Prof. Nicolò Vivona
A QSAR study investigating the potential anti-HIV-1 effect of some Acyclovir and Ganciclovir analogs (NV-3404GP) [pp. 85-94]
Anna Maria Almerico, Marco Tutone and Antonino Lauria
Full Text: PDF (241K)
Supplementary Material: PDF (438K)
N-Methyl-2,6-di-tert-butyl-4,4’-pyrylogen. A dialkyl example of a new class of electron transfer sensitizers (NV-3557GP) [pp. 95-111]
Edward L. Clennan
Full Text: PDF (1,399K)
Supplementary Material: PDF (33K)
Phosphoroamidate derivatives of N,O-nucleosides as inhibitors of reverse transcriptase (NV-3633GP) [pp. 112-124]
Luisa Borrello, Ugo Chiacchio, Antonino Corsaro, Venerando Pistarà and Daniela Iannazzo
Full Text: PDF (310K)
Arkivoc manuscript activity / Traffic at arkat-usa.org

MS in Hand Jan 1st, 2009: 202. Received 71; Published 38; Rejected 51. In Hand End of Jan 184;

Access hits, January: 619,784 from 59,342 visitors;

Individual Issues of Arkivoc
The following issues were completed during January 2009:

2008 Part (i): Special Issue 'Reviews and Accounts'
(Issue completed with 10 papers and 308 pages)

2008 Part (ix): Commemorative Issue in Honor of Prof. Oleg Kulinkovich on the occasion of his 60th anniversary
(Facilitators: Vladimir Tyvorskii and Oleg Epstein; Scientific Editor: Mikael Begtrup)
(Issue completed with 13 papers and 148 pages)

2008 Part (xvi): General Papers
(Issue completed with 30 papers and 326 pages)

No issues were closed during January 2009.
The following new issues were initiated during January 2009:

2008 Part (xvii): General Papers
2010 Part (i): Special Issue 'Reviews and Accounts'
2010 Part (ii): General Papers
2010 Part (iii): Commemorative Issue in Honor of Prof. Benito Alcaide on the occasion of his 60th anniversary
(Facilitator: Pedro Almendros; Scientific Editor: Christopher A. Ramsden)

FloHet 10, U. of Florida, March 8th - 11th, 2009

The Tenth Conference of Heterocyclic and Synthetic Chemistry brochure is at the ARKAT homepage http://www.arkat-usa.org. Registration opened June 2008. Plenary lectures will be given by: Erick Carreira (ETH, Zurich, Switzerland), Janine Cossy (Ecole Superieure de Physique et de Chimie, Paris, France), Frank Fang (Eisai Research Institute, Andover, MA), Ben Feringa (University of Groningen, The Netherlands), Joel Hawkins (Pfizer, New York), Amir Hoveyda (Boston College, MA), Philip Kocienski (University of Leeds, UK), Stephen Martin (University of Texas, Austin, TX), Mike Martinelli (Arena Pharmaceuticals, San Diego, CA), Koji Nakanishi (Columbia University, NY), Chris Senanayake (Boehringer Ingelheim, Germany).

Comprehensive Heterocyclic Chemistry III

Comprehensive Heterocyclic Chemistry III, a new print and online reference work from Elsevier, was recently "RECOMMENDED" by Choice Magazine for being "excellent in general." Visit the website to learn more or to recommend this title to a colleague, and be sure to look for our display at Flohet 2009!

Arkivoc Reached 126 Countries in 2008!

8,046,819 Accesses were recorded to the Arkat website during the year.
(i) From USA 31.9%, Brazil 0.9%, Canada 0.7%, Mexico 0.5%, Argentina 0.3%, and 6.5% from other American Countries.
(ii) From Russia 3.2%, Germany 1.6%, Italy 1.3%, France 1.1%, UK 1.0%, Poland 0.8%, Spain 0.7%, Turkey 0.3%, and 13.1% from other European Countries.
(iii) From India 2.2%, Japan 1.6%, China 0.9%, Indonesia 0.4% and 2.1% from other Asian Countries.
(iv) From Australia 0.4%, and 0.1% from other Pacific Countries.
(v) From Private visitors 28.4%

Online Submission of Arkivoc Manuscripts

Online submission of Arkivoc is now fully operational and will greatly enhance the rate of publication. Authors are strongly encouraged to use the system rather than just submit papers to Dr. Boulton by e-mail. However, the latter method remains the standby in case of system failure.

Additions to Arkivoc Editorial Board of Referees
Nov 2008-Jan 2009

Since November 2008 a total of 19 new referees have been appointed to the Editorial Board of Referees of Arkivoc.

Availability of Printed Arkivoc

We are changing the arrangements for the printed edition for Arkivoc. A limited number of printed copies of all 88 issues covering 2000 – 2007 will be available at the Flohet conferences at $20 per copy. For 2008 issues, printed copies will be produced for Commemorative issues only. From 2009 onwards new arrangements will be made for printed copies as will be detailed in a subsequent newsletter.

To Announce and Advertise in Arkivoc or at FloHet

For details of opportunities on web site, or in Arkivoc, this newsletter, or our conference manual, contact Eric Scriven - Efvs1@aol.com.

New Members
of the Arkivoc Editorial Board of Referees
Prof. Ramesh C. Gupta
India
email
Dr. Joaquin G. Marrero
Spain
email