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MONTHLY NEWSLETTER
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July 31, 2010
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Sent free to the Editorial Board of Referees and any other interested chemists who request it
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ARKIVOC is an international journal of organic chemistry completely free electronically world wide.
No downloading fees to readers and no page or other charges to authors.
Arkat USA, Inc. is a non profit foundation existing to help chemists throughout the world with special emphasis on international cooperation and developing countries.
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Arkivoc manuscript activity / Traffic at arkat-usa.org
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MS in Hand Jul 1st, 2010: 270. Received 137; Published 42; Rejected 114. In Hand End of Jul 251;
Manuscripts in Hand Jan 1st, 2010: 206; Received 773; Published 159; Rejected 568.
Access hits, July: 606,069 from 135,853 visitors;
2010 to date: 4,168,713 from 697,495 visitors.
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Accounts and Reviews Published during July 2010
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Part (i): Special Issue 'Reviews and Accounts'
Gewald reaction: synthesis, properties and applications of substituted 2-aminothiophenes (10-5309LR)
Zita Puterova, Albeta Krutoíková and Daniel Végh
Full Text: PDF (585K) a review with 90 references
pp. 209 - 246
received Apr 15 2010; accepted May 28 2010; published Jul 9 2010.
Three different approaches to C-H bond functionalization in the synthesis of antitumor alkaloids rhazinilam, rhazinal and rhazinicine (10-5425LR)
Delphine Le Floch, Nicolas Gouault, Michčle David and Pierre van de Weghe
Full Text: PDF (720K) a review with 12 references
pp. 247 - 259
received May 20 2010; accepted Jul 2 2010; published Jul 19 2010.
Mechanistic studies of tyrosinase suicide inactivation (10-5374LU)
Christopher A. Ramsden and Patrick A. Riley
Full Text: PDF (462K) an account with 37 references
pp. 260 - 274
received May 5 2010; accepted Jun 17 2010; published Jul 30 2010.
Synthesis and properties of hydrazones bearing amide, thioamide, and amidine functions (10-5215LR)
Nataliya P. Belskaya, Wim Dehaen and Vasiliy A. Bakulev
Full Text: PDF (1,338K) a review with 52 references
pp. 275 - 332
received Mar 16 2010; accepted May 27 2010; published Jul 30 2010.
Part (vii): A Commemorative Issue in Honor of Professor Richard A. Bartsch
Base-promoted elimination reactions of (E)- and (Z)-arylaldehyde O-benzoyloximes. Effects of stereochemistry, ß-aryl group and base-solvent on the nitrile-forming transition states (RB-4931RU)
Sang Yong Pyun and Bong Rae Cho
Full Text: PDF (351K) an account with 38 references
pp. 118 - 137
received Dec 29 2009; accepted Jun 3 2010; published Jul 15 2010.
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Graphical Abstracts
of Manuscripts Published in Arkivoc During July 2010
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Arkivoc 2010 Part (i):
Special Issue 'Reviews and Accounts'
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Gewald reaction: synthesis, properties and applications of substituted 2-aminothiophenes (10-5309LR) [pp. 209-246]
Zita Puterova, Albeta Krutoíková and Daniel Végh
Full Text: PDF (585K)
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Three different approaches to C-H bond functionalization in the synthesis of antitumor alkaloids rhazinilam, rhazinal and rhazinicine
(10-5425LR) [pp. 247-259]
Delphine Le Floch, Nicolas Gouault, Michčle David and Pierre van de Weghe
Full Text: PDF (720K)
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Mechanistic studies of tyrosinase suicide inactivation (10-5374LU) [pp. 260-274]
Christopher A. Ramsden and Patrick A. Riley
Full Text: PDF (462K)
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Synthesis and properties of hydrazones bearing amide, thioamide and amidine functions (10-5215LR) [pp. 275-332]
Nataliya P. Belskaya, Wim Dehaen and Vasiliy A. Bakulev
Full Text: PDF (1,338K)
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Arkivoc 2010 Part (iv):
A Commemorative Issue in Honor of Prof. James Cook
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An enantioselective formal synthesis of (+)-gephyrotoxin 287C (JC-4807FP) [pp. 6-14]
Mark L. Trudell, Lei Miao, Hong Shu, April R. Noble, Steven P. Fournet and Edwin D. Stevens
Full Text: PDF (3,975K)
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An improved synthesis of a ring-C precursor to cobyric acid (JC-4882FP) [pp. 15-24]
Peter Alan Jacobi and Hui Wang
Full Text: PDF (201K)
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Arkivoc 2010 Part (vii):
A Commemorative Issue in Honor of Prof. Richard A. Bartsch
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Metal ion complexation in acetonitrile by upper-rim
benzyl-substituted, di-ionized calix[4]arenes bearing two dansyl fluorophores (RB-5264RU) [pp. 81-97]
Űmmühan Ocak, Miraç Ocak, Xin Shen, Alexander H. Gorman, Kazimierz Surowiec and Richard A. Bartsch
Full Text: PDF (370K)
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Sterically congested, geminal aryl-substituted, proton-ionizable sym-dibenzo-16-crown-5 lariat ethers: synthesis and alkali metal cation extraction
(RB-5067RP) [pp. 98-117]
Chuqiao Tu, Youngchan Jang, Carrie L. Bates, Jerzy Gega, Kazimierz Surowiec and Richard A. Bartsch
Full Text: PDF (353K)
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Base-promoted elimination reactions of (E)- and (Z)-arylaldehyde O-benzoyloximes. Effects of stereochemistry, β-aryl group and base-solvent on the nitrile-forming transition states (RB-4931RU) [pp. 118-137]
Sang Yong Pyun and Bong Rae Cho
Full Text: PDF (351K)
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Synthesis, structure and metal ion binding of di-(1,8-naphtho)-16-crown-4 compounds
(RB-5270RU) [pp. 138-145]
Lokman Torun, Peter Mueller, Xiaodan Cao and Richard A. Bartsch
Full Text: PDF (658K)
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Probing optical recognition of metal ions with employment of
cationic dye-calix[4]arene supramolecular complexes
(RB-5007RP) [pp. 146-159]
Galina G. Talanova, Elena Yu. Vedernikova, Nicole M. Buie, Evan Staunton and Vladimir S. Talanov
Full Text: PDF (311K)
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Effect of Na+ on solvent extraction of alkaline earth metal cations by proton-ionizable calix[4]arenes (RB-4962RP) [pp. 160-169]
Galina G. Talanova, Vladimir S. Talanov, Kazimierz Surowiec and Richard A. Bartsch
Full Text: PDF (256K)
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Arkivoc 2010 Part (viii):
A Commemorative Issue in Honor of Dr. Bruce E. Maryanoff
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Modulation of an n→π* interaction with α-fluoro groups (BM-5071HP) [pp. 251-262]
Amit Choudhary, Charles G. Fry and Ronald T. Raines
Full Text: PDF (424K)
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Arkivoc 2010 Part (ix):
General Papers
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Intramolecular cascade radical cyclizations promoted by samarium diiodide (10-5117OP) [pp. 171-177]
Zhang Hu, Si-dong Li and Peng-zhi Hong
Full Text: PDF (139K)
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An efficient oxidation of 2-pyrazolines and isoxazolines by bis-bromine-1,4-diazabicyclo[2.2.2]octane complex (DABCO-Br2) (10-4311MP) [pp. 178-184]
Davood Azarifar, Kaveh Khosravi and Rahman Ali Veisi
Full Text: PDF (155K)
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Amino acid derivatives. Part 5. Synthesis and anti-HIV activity of new sebacoyl precursor derived thioureido-amino acid and phthalimide derivatives (10-5081MP) [pp. 185-195]
Najim A. Al-Masoudi, Nahed Al-Haidery, Naeem T. Faili and C. Pannecouque
Full Text: PDF (224K)
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Synthesis and antimicrobial activities of novel peptide deformylase inhibitors (10-3973MP) [pp. 196-205]
Ling Yin, Wei-Ren Xu, Zhi-Guo Wang, Da-Tong Zhang, Jiong Jia, Yan-Qing Ge, Yan Li and Jian-Wu Wang
Full Text: PDF (225K)
Supplementary Material: PDF (496K)
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A practical synthesis of a novel PPAR alpha agonist (10-5349KP) [pp. 206-215]
Joel Slade, Hui Liu, Mahavir Prashad and Kapa Prasad
Full Text: PDF (240K)
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Convenient and robust one-pot synthesis of symmetrical and unsymmetrical benzyl thioethers from benzyl halides using thiourea (10-4802SP) [pp. 216-228]
Kevin S. Eccles, Curtis J. Elcoate, Simon E. Lawrence and Anita R. Maguire
Full Text: PDF (230K)
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Organocatalytic asymmetric conjugate addition of cyclic 1,3-dicarbonyl compounds to β,γ-unsaturated α-ketoesters (10-5234UP) [pp. 229-243]
Jin-jia Wang, Jin-hua Lao, Zhi-peng Hu, Rui-Jiong Lu, Shao-zhen Nie, Quan-sheng Du and Ming Yan
Full Text: PDF (420K)
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The synthesis of new thiosubstituted butadienes, butenynes and butatrienes (10-4752CP) [pp. 244-256]
Cemil Ibis and Neslihan Beyazit
Full Text: PDF (282K)
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Experimental and DFT study of 2-ferrocenylpropan-2-ol cyclodimerization products (10-5222HP) [pp. 257-268]
Jasmina Lapić, Mario Cetina, Davor akić, Senka Djaković, Valerije Vrček and Vladimir Rapić
Full Text: PDF (404K)
Supplementary Material: PDF (188K)
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A study of [1]benzofuro[3,2-c]pyridine derivatives (10-5279UP) [pp. 269-281]
Denisa Tarabová, Ján Titi, Naďa Prónayová, Anton Gatial and Albeta Krutoíková
Full Text: PDF (485K)
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A facial synthesis of quinazolino[1,4]benzodiazepine alkaloids via reductive N-heterocyclization of N-(2-nitrobenzoyl)amides: total synthesis of asperlicin C, circumdatin H, and its analogues (10-4137MP) [pp. 282-292]
Naim H. Al-Said, Khaled Q. Shawakfeh, Mohammad I. Ibrahim and Sami H. Tayyem
Full Text: PDF (206K)
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Selective alkylation of aminophenols (10-5213GP) [pp. 293-299]
Jiaxi Xu and Renchao Wang
Full Text: PDF (104K)
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Microwave-assisted one-pot reactions for direct synthesis of 6-methylpurines (10-4832OP) [pp. 300-307]
Hai-Ming Guo, Zhi-Jie Mao, Hong-Ying Niu, Dong-Chao Wang, Gui-Sheng Zhang and Gui-Rong Qu
Full Text: PDF (288K)
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Nucleophilic substitution reactions, molecular aggregation, structure and lipophilicity of 6-chloro-3-chloromethyl-1,2,4-triazolo[4,3-b]pyridazine
(10-5347HP) [pp. 308-318]
Anna Katrusiak and Andrzej Katrusiak
Full Text: PDF (445K)
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Microwave-assisted C-C cross-coupling reactions of aryl and heteroaryl halides in water (10-5361DP) [pp. 319-330]
Kamal M. Dawood and Moteaa M. El-Deftar
Full Text: PDF (225K)
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Arkivoc 2010 Part (x):
General Papers
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Synthesis of new calix[4]arenes bearing silylether groups (10-4898BP) [pp. 1-10]
Kazem D. Safa and Yones Mosaei Oskoei
Full Text: PDF (380K)
Supplementary Material: PDF (388K)
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On the synthesis of N-maleoyl amino acids in aqueous media: cautionary tales for the unwary traveller (10-5324EP) [pp. 11-16]
Michael John Paterson and Aleksandar Jovanovic
Full Text: PDF (152K)
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Efficient conjugate addition of carbonyl compounds to
3-nitro-2H-chromenes in the presence of bases
(10-5342YP) [pp. 17-33]
Zhi-peng Hu, Jun-min Zhang, Chun-liang Lou, Jin-jia Wang, Shao-zhen Nie,and Ming Yan
Full Text: PDF (341K)
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Flash vacuum pyrolysis of 1,2,5-oxadiazole 2-oxides and 1,2,3-triazole 1-oxides
(10-5281UP) [pp. 34-54]
William R. Mitchell and R. Michael Paton
Full Text: PDF (365K)
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A facile asymmetric synthesis of (S)-duloxetine (10-4508EP) [pp. 55-61]
Kee-In Lee, Se Hun Kwak and Jung Min Seo
Full Text: PDF (221K)
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Experimental and theoretical investigation of the structure and nucleophilic properties of 4-aminocoumarin (10-5152QP) [pp. 62-76]
Emil Popovski, Bistra Stamboliyska, Voislava Janevska, Boris Shivachev, Rosica P. Nikolova, Goran Stojkovic and Bozhna Mikhova
Full Text: PDF (522K)
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Stereospecific synthesis of N-tosyl derivatives of dihydroconduramine E-2 and ent-F-2 (10-4817MP) [pp. 77-85]
Izzet N. Kurbanoglu, Senol Besoluk and Mustafa Zengin
Full Text: PDF (164K)
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Reactivity of some structural analogs of dehydroacetic acid DHA with o-phenylenediamine (10-5269EP) [pp. 86-97]
Nabila Ait-Baziz, Yahia Rachedi and Artur M. S. Silva
Full Text: PDF (196K)
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Iodine-promoted facile synthesis of new (+)-2,3-dihydro-N,2-diarylquinazolines
(10-5319BP) [pp. 98-109]
Kamal M. El-Shaieb, Henning Hopf and Peter G. Jones
Full Text: PDF (333K)
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A rapid and simple one-pot procedure for the synthesis of 3β-acetoxy-5α-hydroxy-6-oxo steroids (10-5377BP) [pp. 110-115]
Anielka Rosado-Abón, Margarita Romero-Ávila and Martin A. Iglesias-Arteaga
Full Text: PDF (246K)
Supplementary Material: PDF (901K)
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Synthesis of aminopyrrolo[1,2-a]thieno[3,2-e]pyrazine derivatives as serotoninergic 5-HT7 ligands
(10-5069VP) [pp. 116-131]
Grégoire Pavé, Saďd Lazar, Aurélien Lesnard, Sylvain Rault and Gérald Guillaumet
Full Text: PDF (182K)
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Regioselective transformation of 6/5-fused bicyclic isoxazolidines to second-generation cyclic aldonitrones
(10-5267QP) [pp. 132-148]
Basem A. Moosa and Shaikh A. Ali
Full Text: PDF (260K)
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Gas-phase pyrolysis of N-alkoxyphthalimides to functionally substituted aldehydes: kinetic and mechanistic study (10-4997OP) [pp. 149-162]
Alya M. Al-Etaibi, Nouria A. Al-Awadi, Maher R. Ibrahim and Yehia A. Ibrahim
Full Text: PDF (135K)
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Synthesis and biological evaluation of new indazole derivatives (10-5004EP) [pp. 163-177]
Salvatore Plescia, Demetrio Raffa, Fabiana Plescia, Giovanni Casula, Benedetta Maggio, Giuseppe Daidone, Maria Valeria Raimondi, Maria Grazia Cusimano, Gabriella Bombieri and Fiorella Meneghetti
Full Text: PDF (513K)
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Individual Issues of Arkivoc
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The following issues were completed during July 2010:
2010 Part (v): Commemorative Issue in Honor of Prof. Antonio Rocha-Gonsalves on the occasion of his 70th anniversary
(Facilitator: Teresa M. V. D. Pinho e Melo; Scientific Editor: John A. Joule)
(Issue completed with 15 papers and 182 pages)
2010 Part (ix): General Papers
(Issue completed with 30 papers and 330 pages)
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No issues were closed during July 2010.
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No new issues were initiated during July 2010.
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Flohet 12 to take place at University of Florida Gainesville March 6-9, 2011. Registration now Open
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12th Florida Heterocyclic and Synthetic Conference March 6-9, 2011, University of Florida, Gainesville. Plenary lecturers will include, Jacqueline Barton, Daniel Comins, Francois Diederich, John Hartwig, Yoshito Kishi, Jeffrey Kuethe, Max Malacria, Lieven Meerpoel, George Moniz, Victor Snieckus, and Dinesh Vyas. Registration: www.arkat-usa.org
The 11th Annual Florida Heterocyclic and Synthetic Conference (FloHet-11) took place at the University of Florida in Gainesville, March 7-10. There were 11 plenary lectures, 37 invited lectures, 50 posters, 5 courses, and exposition that attracted 12 exhibitors.
We are most grateful for the generous support of our sponsors, exhibitors, and advertisers AlfaAesar, Bristol-Myers Squibb, CEM, Elsevier, Georg Thieme Verlag KG, IUPAC, MolCode, Oakwood Products, Royal Society of Chemistry, SigmaAldrich, Strem, Synthonix, Taylor & Francis, Vertellus, and The Alachua County Visitors and Convention Bureau.
Some comments from those who attended:
- I am very glad that I attended this conference
- I will strongly encourage my colleagues to attend
- Enabled one to meet people from all over the world
- I made new contacts and enjoyed the chemistry
- Talks were excellent, the poster were great and the mini-courses were fantastic
- Meeting was one of the best I have had the privilege of attending in many years
12th Florida Heterocyclic and Synthetic Conference March 6-9, 2011, University of Florida, Gainesville. Plenary lecturers will include, Jacqueline Barton, Daniel Comins, Francois Diederich, John Hartwig, Yoshito Kishi, Jeffrey Kuethe, Max Malacria, Lieven Meerpoel, George Moniz, Victor Snieckus, and Dinesh Vyas.
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To Announce and Advertise in Arkivoc or at FloHet
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For details of opportunities on web site, or in Arkivoc, this newsletter, or our conference manual, contact Eric Scriven - Efvs1@aol.com.
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Forthcoming Conferences
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45th Congress of the Mexican Chemical Society
29th National Congress of Chemical Education, September 18-22, 2010
Information: www.sqm.org.mx Registration: soquimex@prodigy.net.mx
The 11th Eurasia Conference on Chemical Sciences
Venue: The King Hussain Conference Centre, Dead Sea, Jordan, October, 6 to 10, 2010. Information and registration http://www.euasc2s-11.ju.edu.jo/
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ARKIVE
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ARKIVE is an in-house chemical database of more than 30,000 compounds synthesized by the Prof. Katritzkys research group Department of Chemistry, University of Florida, Gainesville, Florida, USA. These compounds include 1) Lead Generation, 2) Focused Sets, 3) Building Blocks and 4) Reagents for Heterocycle Assisted Syntheses. We have compiled downloadable lists of these chemicals that are updated quarterly. A recent article (J. Chem. Inf. Model 2010, 50, 470-479) by Chuprina et.al. analyses commercially available data bases of compounds from 29 suppliers worldwide, including ours. They concluded that our database of compounds (#28,881) possesses i) 21418 exclusive compounds (74.2%) and ii) 7670 drug-like compounds (26%). Our Arkive database includes both the chemical structure and the identification number for every compound. This database can be downloaded in SD or ISIS format to your local database. You may also access this database at www.ark.chem.ufl.edu. Your inquiries and orders can be addressed to ARKIVE manager Dr. Srinivasa R. Tala by email compounds@chem.ufl.edu or by Fax at 352-392-9199.
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